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Hirokuni Taguchi Selected Research

Phosphotransferases (Kinase)

9/2007AZD1152, a novel and selective aurora B kinase inhibitor, induces growth arrest, apoptosis, and sensitization for tubulin depolymerizing agent or topoisomerase II inhibitor in human acute leukemia cells in vitro and in vivo.
6/2007A novel treatment strategy targeting Aurora kinases in acute myelogenous leukemia.
7/2005HIV-1 protease inhibitor induces growth arrest and apoptosis of human prostate cancer LNCaP cells in vitro and in vivo in conjunction with blockade of androgen receptor STAT3 and AKT signaling.

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Hirokuni Taguchi Research Topics

Disease

25Neoplasms (Cancer)
02/2008 - 08/2002
10Prostatic Neoplasms (Prostate Cancer)
09/2007 - 10/2003
10Lung Neoplasms (Lung Cancer)
04/2007 - 06/2002
8Leukemia
09/2007 - 12/2003
6Adult T-Cell Leukemia-Lymphoma (Leukemia Lymphoma, T Cell, Acute, HTLV I Associated)
02/2008 - 06/2003
5Acute Myeloid Leukemia (Acute Myelogenous Leukemia)
09/2007 - 08/2002
5Lymphoma (Lymphomas)
06/2007 - 12/2002
5Non-Small-Cell Lung Carcinoma (Carcinoma, Non-Small Cell Lung)
03/2007 - 02/2003
5Multiple Myeloma
10/2006 - 02/2004
5Myeloid Leukemia (Leukemia, Myelocytic)
08/2006 - 10/2003
4Precursor Cell Lymphoblastic Leukemia-Lymphoma (Acute Lymphoblastic Leukemia)
09/2007 - 12/2002
4BCR-ABL Positive Chronic Myelogenous Leukemia (Chronic Myelogenous Leukemia)
09/2007 - 08/2002
3Small Cell Lung Carcinoma (Small Cell Lung Cancer)
09/2007 - 05/2003
3Hematologic Neoplasms (Hematological Malignancy)
10/2006 - 02/2004
2Hypereosinophilic Syndrome (Loeffler Endocarditis)
03/2009 - 10/2006
2Eosinophilia
03/2009 - 01/2007
2Blast Crisis (Blast Phase)
09/2007 - 10/2006
2Ocular Paraneoplastic Syndromes
09/2007 - 06/2007
2Non-Hodgkin Lymphoma (Lymphosarcoma)
10/2006 - 04/2005
2Neoplasm Metastasis (Metastasis)
08/2006 - 03/2006
2Idiopathic Thrombocytopenic Purpura (Thrombocytopenic Purpura, Autoimmune)
11/2005 - 11/2002
2Thrombocytopenia (Thrombopenia)
11/2005 - 11/2002
2Epstein-Barr Virus Infections
05/2005 - 05/2003
2Acute Promyelocytic Leukemia
10/2003 - 10/2003
1Chronic Cough
03/2009
1Cough
03/2009
1Asthma (Bronchial Asthma)
03/2009
1Acute Eosinophilic Leukemia
09/2007
1Burkitt Lymphoma (Burkitt's Lymphoma)
06/2007
1Diffuse Large B-Cell Lymphoma (Lymphoma, Large Cell, Diffuse)
06/2007
1Carcinogenesis
06/2007
1Aneuploidy (Aneuploid)
06/2007
1Thrombosis (Thrombus)
01/2007
1Sarcoma (Soft Tissue Sarcoma)
01/2007
1Gastrointestinal Stromal Tumors (Gastrointestinal Stromal Tumor)
09/2006

Drug/Important Bio-Agent (IBA)

8NF-kappa B (NF-kB)IBA
02/2008 - 12/2003
8Biological ProductsIBA
06/2007 - 06/2002
6herbal preparation PC-SPESIBA
09/2007 - 10/2003
6AndrogensIBA
09/2007 - 11/2003
6DNA (Deoxyribonucleic Acid)IBA
06/2007 - 12/2002
5Proteins (Proteins, Gene)FDA Link
09/2007 - 02/2004
5Granulocyte Colony-Stimulating Factor (G-CSF)IBA
04/2007 - 06/2002
5Granulocyte-Macrophage Colony-Stimulating Factor (GM-CSF)IBA
04/2007 - 02/2003
4Androgen Receptors (Androgen Receptor)IBA
09/2007 - 11/2003
4Human immunodeficiency virus 1 p16 proteaseIBA
08/2006 - 04/2004
3Imatinib Mesylate (Gleevec)FDA Link
03/2009 - 08/2002
3Adrenal Cortex Hormones (Corticosteroids)IBA
03/2009 - 12/2002
3Phosphotransferases (Kinase)IBA
09/2007 - 07/2005
3Ritonavir (Norvir)FDA Link
08/2006 - 04/2004
3Complementary DNA (cDNA)IBA
08/2006 - 08/2002
3Tretinoin (Retinoic Acid)FDA LinkGeneric
10/2004 - 04/2004
2ThymidineIBA
09/2007 - 06/2007
2Aurora KinasesIBA
09/2007 - 06/2007
2RecoverinIBA
09/2007 - 06/2007
2TOR Serine-Threonine KinasesIBA
05/2007 - 10/2006
2Sirolimus (Rapamycin)FDA Link
05/2007 - 10/2006
2Cyclooxygenase 2 (Cyclooxygenase-2)IBA
04/2007 - 08/2004
2Sunitinib (Sutent)FDA Link
10/2006 - 09/2006
2Calcitriol (Calcijex)FDA LinkGeneric
08/2006 - 06/2005
2Trypan BlueFDA Link
06/2006 - 10/2003
2Nelfinavir (Viracept)FDA Link
07/2005 - 04/2004
2oridoninIBA
04/2005 - 10/2003
2Indinavir (Crixivan)FDA Link
10/2004 - 04/2004
2Saquinavir (Invirase)FDA Link
10/2004 - 04/2004
2Pharmaceutical PreparationsIBA
10/2004 - 10/2004
2SteroidsIBA
09/2004 - 08/2003
2Cyclooxygenase 2 Inhibitors (COX-2 Inhibitors)IBA
08/2004 - 02/2003
2Proteasome InhibitorsIBA
03/2004 - 02/2004
2Prostate-Specific Antigen (Semenogelase)IBA
03/2004 - 11/2003
2Bortezomib (Velcade)FDA Link
03/2004 - 02/2004
1Topoisomerase II InhibitorsIBA
09/2007
12- ((3- ((4- ((5- (2- ((3- fluorophenyl)amino)- 2- oxoethyl)- 1H- pyrazol- 3- yl)amino)quinazolin- 7- yl)oxy)propyl)(ethyl)amino)ethyl dihydrogen phosphateIBA
09/2007
14- (4- (N- benzoylamino)anilino)- 6- methoxy- 7- (3- (1- morpholino)propoxy)quinazolineIBA
09/2007
1Aurora Kinase BIBA
09/2007
1TubulinIBA
09/2007
1saw palmetto extractIBA
09/2007
1BromidesIBA
09/2007
1AutoantibodiesIBA
09/2007
1Retinaldehyde (Retinal)IBA
09/2007
1Bone Morphogenetic Protein 6IBA
06/2007
1Annexin A5IBA
06/2007
1Aurora Kinase AIBA
06/2007
1Phosphatidylinositol 3-Kinase (1 Phosphatidylinositol 3 Kinase)IBA
05/2007
12- (4- morpholinyl)- 8- phenyl- 4H- 1- benzopyran- 4- oneIBA
05/2007
1Granulocyte-Macrophage Colony-Stimulating Factor Receptors (GM-CSF Receptor)IBA
04/2007
1Granulocyte Colony-Stimulating Factor Receptors (G-CSF Receptor)IBA
04/2007
1Histones (Histone)IBA
03/2007
1Tumor Biomarkers (Tumor Markers)IBA
01/2007
1Protein-Tyrosine Kinases (Tyrosine Kinase)IBA
10/2006
1Peptide Initiation Factors (Initiation Factor)IBA
10/2006
170-kDa Ribosomal Protein S6 Kinases (Ribosomal Protein S6 Kinases, 70 kDa)IBA
10/2006
1Receptor Protein-Tyrosine Kinases (Tyrosine Kinase Receptors)IBA
10/2006
1EverolimusFDA Link
10/2006
1Macrophage Colony-Stimulating FactorIBA
08/2006
1Colony-Stimulating Factors (Colony Stimulating Factor)IBA
08/2006
1Dinoprostone (PGE2)FDA Link
08/2006
1Transcription Factors (Transcription Factor)IBA
08/2006

Therapy/Procedure

12Therapeutics
01/2007 - 09/2003
3Drug Therapy (Chemotherapy)
12/2003 - 08/2002
1Pneumonectomy (Lung Volume Reduction)
01/2007